Anti Estrogen PCT Tamoxifen Citrate Nolvadex CAS 54965-24-1 Tamoxifen Raw Powder

 

Tamoxifen Citrate

 

 

Quick Details:

Product Name: Tamoxifen Citrate

Synonyms: Tamoxifen , Nolvadex

CAS: 54965-24-1

MF: C32H37NO8

MW: 563.64

EINECS: 259-415-2

Melting point: 140-144 °C

storage temp: 2-8°C

solubility  methanol: soluble50mg/mL, clear, colorless

Water Solubility: slightly soluble

Stability: Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months

 

 

 

 

COA :

Test Items	Analysis Standard	Results
Identification	Conform	Conform
Heavy metals	0.001%	Conform
Specific Rotation	﹢34°~﹢40°	+36.3°
Chromatography Purity	Conform	Conform
Melting point	142~ 148℃	144~148℃
Organic Volatile Impurities	Conform	Conform
Loss On Drying	≤0.5%	0.15%
Residue On Ignition	0.2%max	0.08%
Assay	98.0%min	99.58%

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

Description:

Nolvadex is an estrogen agonist in the liver, capable of activating the estrogen receptor and mimicking the actions of this sex hormone in this region of the body. As such it can have a markedly positive impact on HDL (good) cholesterol values, as does estrogen. Many similarly use this drug to counter some of the negative consequences of steroid use in regards to cholesterol values and cardiac risk, as steroids often suppress HDL and raise LDL levels considerably. in some instances an athlete is able to maintain a very favorable HDL/LDL cholesterol ratio, to spite the use of a mode rate dosage (400mg weekly) of an injectable like testosterone or nandrolone. It would be foolish to think however that Nolvadex would be a sufficient remedy with the heavy use of c-l7alpha alkylated orals or extremely high dosed cycles in general

 

The drug is technically an estrogen agonist/antagonist, which competitively binds to estrogen receptors in various target tissues. With the tamoxifen molecule bound to this receptor, estrogen is blocked from exerting any action, and an anti-estrogenic effect is achieved. Since many forms of breast cancer are responsive to estrogen, the ability of tamoxifen citrate to block its action in such cells has proven to be a very effective treatment.

 

It is also utilized successfully as a preventative measure, taken by people with an extremely high familial tendency for breast cancer. While Nolvadex is effective against estrogen, it is not our strongest available remedy. We now have the drugs Arimidex, Femara, and Aromasin available to us, which notably prevents estrogen from being manufactured in the first place. Altering the effect of estrogen in the female body can cause a level of discomfort, so anti-estrogens are most bearable when used after the point of menopause. Since Nolvadex is milder in comparison, it is more widely applicable and usually the first treatment option.

 

 

Application:

The claim that Nolvadex reduces gains should not be taken too seriously. The fact is that any number of bodybuilders have made excellent gains while using Nolvadex. The belief that it reduces gains seems to stem from the fact that the scientific literature reports a slight reduction in IGF-1 (individuals using anabolic steroids were not studied though) from use of Nolvadex.

 

Tamoxifen slows or stops the growth of cancer cells that are already present in the body. It helps keep the original breast cancer from coming back and helps prevent new cancer in the opposite breast. It also reduces the risk of breast cancer in women who have a high risk for this disease.

 

Tamoxifen is highly effective in lowering the risk of breast cancer recurrence. In women who have already had breast cancer, tamoxifen also lowers the risk of breast cancer in the opposite breast (contralateral).Tamoxifen is used to prevent and treat breast cancers that test positive for estrogen receptors (ER+). It blocks the effects that the hormone estrogen has on cancer cells and lowers the chance that breast cancer will grow. It is often called an "anti-estrogen."For postmenopausal women, a two-stage treatment using tamoxifen and then an aromatase inhibitor, such as anastrozole (Arimidex), exemestane (Aromasin), or letrozole (Femara) may work better than only taking tamoxifen.

 

 

What we supply is Tamoxifen Citrate oral raw :

1. Tamoxifen Citrate is a SERM that acts as both antagonist and agonist in relation to the estrogen hormone. It is an anti-estrogen in that it binds to estrogen receptors in certain parts of the body, particularly in the mammary tissue. This action prevents estrogen from acting on its originally intended point of binding.

 

2. Tamoxifen Citrate acts as an estrogen on the liver. Liver related estrogenic activity has been shown to improve cardiovascular health, particularly as it relates to cholesterol. This can be very advantageous for the bodybuilding steroid user as most steroids have a negative impact on cholesterol levels.

 

3. Beyond its estrogen related activity Tamoxifen Citrate possesses strong testosterone stimulating properties. The use of Tamoxifen Citrate will stimulate the pituitary to increase its production of Luteinizing Hormone (LH) and Follicle Stimulating Hormone (FSH) with a strong emphasis on LH. LH and FSH are the gonadotropins that signal to the testicles to produce testosterone. Without LH and FSH there is no testosterone production.

 

 

What is the usual dosage ?
The information below is based on the dosage guidelines your doctor uses. Depending on your condition and medical history, your doctor may prescribe a different regimen. Do not change the dosage or stop taking your medication without your doctor's approval.

1. Breast Cancer Treatment

The usual dosage ranges from 20-40 milligrams (mg) daily. If you are taking >20 mg a day, your doctor will have you divide the total into two smaller doses taken in the morning and evening.

 

2. Ductal Carcinoma in Situ

The usual dose is 20 mg daily for 5 years.

 

3. To Reduce the Incidence of Breast Cancer in High-Risk Women
The usual dose is 20 mg daily for 5 years.